σ1 Receptor/μ Opioid receptor modulator 2 - CAS 3009018-61-2

Compound 4x, also known as σ1 Receptor/μOpioid receptormodulator 2, acts as a μOR agonist and a σ1R antagonist, exhibiting a potent μOR EC50 of 0.6 nM and strong σ1R inhibitory activity (Ki: 363.7 nM) . It demonstrates significant analgesic effects in various pain models.

Sigma receptor, Opioid Receptor

Endocrinology/Hormones, Neuroscience, GPCR/G Protein

3008955

C23H31N3O

365.51

O=C(N(C1=NC=CC=C1)CC(N2CCC(C=3C=CC=CC3)CC2)CC)CC

-20°C

Ice Packs

Small Compound