β3-AR agonist 1 - CAS 1283125-73-4

β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold) .

Others, Adrenergic Receptor

Others, GPCR/G Protein, Neuroscience

1283048

C22H28N4O4S

444.55

CC=1C=2C(=CC(OCCNC[C@H](O)C3=CC(NS(=O)(=O)C4CCC4)=CC=C3)=CC2)NN1

-20°C

Ice Packs

Small Compound