3-IN-PP1 - CAS 2227110-54-3

3-IN-PP1, a potent protein kinase D (PKD) inhibitor, exhibits pan-PKD inhibitory activity with IC50 values of 108 nM for PKD1, 94 nM for PKD2, and 108 nM for PKD3. Additionally, it serves as a broad-spectrum anticancer agent by inhibiting the growth of various tumor cells. 3-IN-PP1 is utilized in cancer research [1].

Others, Serine/threonin kinase

Metabolism, Cell Cycle/Checkpoint, Others

2227053

C17H18N6

306.36

NC1=C2C(=NN(C(C)(C)C)C2=NC=N1)C=3C=4C(NC3)=CC=CC4

-20°C

Ice Packs

Small Compound