5-HT2A/5-HT2C inverse agonist 1 - CAS 2718990-76-0

5-HT2A/5-HT2C inverse agonist 1 serves as a dual and potent inverse agonist for the 5-HT2A and 5-HT2C receptors, with hERG inhibition properties that mitigate cardiovascular risks. Demonstrating significant antipsychotic efficacy in the MK-801-induced mouse model, this compound holds potential for psychosis research.

5-HT Receptor

Neuroscience, GPCR/G Protein

2718914

C24H35N5O2

425.57

N(CC1=NN(C)C=C1)(C(NCC2=CC=C(OCCC)C=C2)=O)[C@@H]3C4(CC4)CN(C)CC3

-20°C

Ice Packs

Small Compound