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5-HT2CR agonist 1 - CAS 1216074-15-5

5-HT2CR agonist 1 - CAS 1216074-15-5

MF-0059517-01

$1,383.80 USD
$1,383.80 USD
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Product Details

  • Bioactivity

    The compound 5-HT2CR agonist 1 (compound 8), a 7-chloro analogue, is a selective partial agonist for the 5-HT2C receptor, exhibiting an Emax of 71.09% and an EC50 of 121.5 nM, with no activity observed toward 5-HT2A or 5-HT2B receptors. It does not recruit β-arrestin and shows low hERG inhibition at 10 μM [1].

  • Target

    5-HT Receptor

  • Related Pathways

    GPCR/G Protein, Neuroscience

  • CAS Number

    1216074-15-5

  • Molecular Formula

    C13H14ClNO

  • Molecular Weight

    235.71

  • SMILES

    ClC=1C=CC=2C=CC3(OC2C1)CCNCC3

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound