Ac-RYYRWK-NH2 TFA - CAS 408305-09-9

Ac-RYYRWK-NH2 is a highly effective and specific partial agonist for the nociceptin receptor (NOP) . It demonstrates a remarkable affinity for rat cortical membranes ORL1, with [3H]Ac-RYYRWK-NH2 exhibiting a Kd value of 0.071 nM. However, it shows negligible affinity towards μ-, κ-, or δ-opioid receptors.

Opioid Receptor

Endocrinology/Hormones, Neuroscience, GPCR/G Protein

408305-09-9

C51H70F3N15O11

1126.21

OC(=O)C(F)(F)F.CC(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CCCCN)C(N)=O

-20°C

Ice Packs

Peptide