Adenosine receptor inhibitor 1 - CAS 2550400-52-5

Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR), exhibiting exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >1000, >1000 nM. This compound demonstrates notable antinociceptive, anti-inflammatory, and peripheral analgesic properties, holding great promise for investigating cancer and neurodegenerative diseases [1].

Adenosine Receptor, Others

GPCR/G Protein, Others, Neuroscience

2550343

C17H19ClFN5O3

395.82

CN1C2=C(N(C)C(NCC3=C(F)C(OC)=CC=C3Cl)=N2)C(=O)N(CC)C1=O

-20°C

Ice Packs

Small Compound