AM841 - CAS 871978-21-1

AM841, a high-affinity electrophilic ligand, covalently interacts with a cysteine residue in helix six, thus activating the CB1 cannabinoid receptor. It diminishes forskolin-stimulated cAMP accumulation and slows gastrointestinal motility [1] [2].

Cannabinoid Receptor

GPCR/G Protein

871956

C26H39NO3S

445.66

OC1=C2[C@]3([C@](C(C)(C)OC2=CC(C(CCCCCCN=C=S)(C)C)=C1)(CC[C@@H](CO)C3)[H])[H]

-20°C

Ice Packs

Small Compound