Molfinity

Antihistamine-1 - CAS 1186430-60-3

SKU:MF-0004423-01

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Size 100 mg 5 mg 1 mL - 10 mM (in DMSO) 10 mg 25 mg 50 mg

Product Details

Bioactivity
Antihistamine-1 is an H1-antihistamine (Ki: 6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel (IC50s: 5.4 and 0.8 μM) .
Target
Cytochromes P450, Potassium Channel, Histamine Receptor
Related Pathways
GPCR/G Protein, Immunology/Inflammation, Neuroscience, Membrane transporter/Ion channel, Metabolism
CAS Number
1186367
Purity
>99.99%
Molecular Formula
C23H24FN5
Molecular Weight
389.47
SMILES
C(N1C(=NC=2C1=CC=CC2)N3CCC(CC3)N4C=C(C)C=N4)C5=CC=C(F)C=C5
Storage Temperature
-20°C
Shipping Conditions
Ice Packs
Category
Small Compound