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Molfinity

Antitumor agent-101 - CAS 2848632-52-8

Antitumor agent-101 - CAS 2848632-52-8

SKU:MF-0147102-01

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  • Bioactivity

    Antitumor agent-101 is a selective, covalent inhibitor targeting lysine methyltransferases G9a/GLP, demonstrating IC50 values of 8.5 nM for G9a and 5.5 nM for GLP. It exhibits antitumor efficacy in the PANC-1 xenograft model [1].

  • Target

    Histone Methyltransferase, Glucagon Receptor

  • Related Pathways

    GPCR/G Protein, Chromatin/Epigenetic

  • CAS Number

    2848572

  • Molecular Formula

    C26H38N6O3

  • Molecular Weight

    482.62

  • SMILES

    N(C=1C2=C(C=C(OCCCN3CCCC3)C(OC)=C2)N=C(N(C(C=C)=O)C)N1)C4CCN(C)CC4

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound