APC-6860 - CAS 154628-42-9

APC-6860 is a trypsin-like serine protease inhibitor with \ (k_i \) values of 0.21, 0.44, 1.5, 16.8, 20, and 30 μM for uPA, trypsin, tryptase, tPA, thrombin, and factor Xa, respectively. It exhibits a selectivity ratio for tPA versus uPA of 80 and has \ (k_i \) values of 0.1 and 0.082 μM for human and murine urokinases, respectively. APC-6860 can be utilized for cancer research.

Others, Serine Protease

Proteases/Proteasome, Others

154577

C9H7IN2S

302.13

NC(=N)c1cc2c(I)cccc2s1

-20°C

Ice Packs

Small Compound