Bilaid C - CAS 2393866-13-0

Bilaid C is a tetrapeptide μ-opioid receptor agonist (Ki= 210 nM in HEK293 cell membranes expressing the human receptor) that has been found inPenicillium.1It inhibits forskolin-induced cAMP accumulation by 77% in HEK293 cells expressing the human μ-opioid receptor when used at a concentration of 10 μM. Bilaid C induces inward rectifying potassium channel (Kir) currents in rat locus coeruleus slices that endogenously express high levels of the μ-opioid receptor (EC50= 4.2 μM) .

Opioid Receptor

Neuroscience, Endocrinology/Hormones, GPCR/G Protein

2393866-13-0

C28H38N4O6

526.62

CC(C)[C@H](NC(=O)[C@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(C)C)C(=O)N[C@H](Cc1ccccc1)C(O)=O

-20°C

Ice Packs

Peptide