BMS-248360 - CAS 254737-87-6

BMS-248360 is a potent, orally active dual antagonist of both angiotensin II receptor (AT1) and endothelin A (ETA) receptor, with Kis of 10 nM and 1.9 nM for hAT1 and hETA receptors, respectively. BMS-248360 demonstrates hypertensive effects[1].

Endothelin Receptor, RAAS, Others

GPCR/G Protein, Endocrinology/Hormones, Others

254644

C36H45N5O5S

659.84

O=C1C2(N=C(CCCC)N1CC3=CC(CN4C(=O)C(C)(C)CC4)=C(C=C3)C5=C(S(NC6=C(C)C(C)=NO6)(=O)=O)C=CC=C5)CCCC2

-20°C

Ice Packs

Small Compound