Bombinakinin M - CAS 509151-65-9

Potent bradykinin receptor agonist. Highly selective for mammalian arterial smooth muscle bradykinin receptors, displaying ~ 50-fold greater potency than bradykinin. Elicits dose-dependent contractile effects in smooth muscle of guinea pig ileum (EC50 = 4.0 nM) .

Bradykinin Receptor

GPCR/G Protein

509151-65-9

C100H159N31O24

2179.55

C(=O)([C@H]1N(C([C@@H](NC(=O)[C@H]2N(C(CNC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC(=O)[C@H]3N(C([C@@H](NC([C@H](CC(O)=O)N)=O)CC(C)C)=O)CCC3)CCCCN)=O)[C@H](CC)C)=O)CC(N)=O)=O)CCCNC(=N)N)=O)CCCCN)=O)=O)CCC2)CCCNC(=N)N)=O)CCC1)N4[C@H](C(NCC(N[C@@H](CC5=CC=CC=C5)C(N[C@H](C(=O)N6[C@H](C(N[C@@H](CC7=CC=CC=C7)C(N[C@@H](CCCNC(=N)N)C(O)=O)=O)=O)CCC6)CO)=O)=O)=O)CCC4

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