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Molfinity

Brilaroxazine - CAS 1239729-06-6

Brilaroxazine - CAS 1239729-06-6

SKU:MF-0016892-01

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  • Bioactivity

    Brilaroxazine (RP5063) is a potent multimodal dopamine/5-HT modulator. Brilaroxazine is a partial agonist of dopamine D2, D3, and D4 receptors, 5-HT1A (Ki =1.5 nM) and 5-HT2A (Ki = 2.5 nM), and has antagonist activity 5-HT2B, and 5-HT7 receptors with Kis of 0.19 nM and 2.7 nM, respectively. Brilaroxazine can be used for research about cognitive impairments in neuropsychiatric and neurological diseases.

  • Target

    Dopamine Receptor, 5-HT Receptor

  • Related Pathways

    GPCR/G Protein, Neuroscience

  • CAS Number

    1239729-06-6

  • Purity

    0.9936

  • Molecular Formula

    C22H25Cl2N3O3

  • Molecular Weight

    450.36

  • SMILES

    Clc1cccc(N2CCN(CCCCOc3ccc4OCC(=O)Nc4c3)CC2)c1Cl

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound