BRK inhibitor P21d hydrochloride - CAS 2250025-98-8

BRK inhibitor P21d hydrochloride is a highly potent inhibitor of breast tumor kinase (BRK/PTK6), displaying an IC50 of 30 nM, and effectively suppresses p-SAM68 with an IC50 of 52 nM. This compound serves as a valuable tool for evaluating BRK inhibitors' efficacy in xenograft breast tumor models, enabling in vivo activity assessment.

Others, BTK

Tyrosine Kinase/Adaptors, Angiogenesis, Others

2249919

C23H23ClFN7O2

483.93

Cl.Fc1cc(ccc1Nc1nc(cn2c(cnc12)-c1cn[nH]c1)C1CC1)C(=O)N1CCOCC1

-20°C

Ice Packs

Small Compound