Bromodomain IN-2 - CAS 2445335-77-1

BD-IN-1, a pan bromodomain (BD) inhibitor, exhibits K_D values of 250 nM for BRD4 (1), 420 nM for CBP, 130 nM for BRPF1B, 430 nM for BRD7, 67 nM for BRD9, 240 nM for BRDT (1), and 970 nM for CECR2, respectively. This compound demonstrates antiproliferative activity [1].

Epigenetic Reader Domain, Others

Chromatin/Epigenetic, Others

2445257

C16H17ClN2O

288.77

ClC1=C(C2=C3C(=C(C)N2)C(=O)CCCC3)C=C(N)C=C1

-20°C

Ice Packs

Small Compound