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Molfinity

BX-912 - CAS 702674-56-4

BX-912 - CAS 702674-56-4

SKU:MF-0094620-01

Regular price $45.88 USD
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  • Bioactivity

    BX-912 is a specific inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1, IC50: 12 nM) . The selectivity of BX-912 is more 10 fold than C-Kit, EGFR, PKA, PKC etc.

  • Target

    PKA, PDK, Chk, VEGFR, Apoptosis, CDK

  • Related Pathways

    Angiogenesis, Apoptosis, PI3K/Akt/mTOR signaling, Tyrosine Kinase/Adaptors, Cell Cycle/Checkpoint

  • CAS Number

    702614

  • Purity

    0.9934

  • Molecular Formula

    C20H23BrN8O

  • Molecular Weight

    471.35

  • SMILES

    Brc1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCc1cnc[nH]1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound