CAY10771 - CAS 2522599-79-5

CAY10771 is a dual agonist of farnesoid X receptor (FXR) and peroxisome proliferator-activated receptor δ (PPARδ) .1It activates FXR and PPARδ in reporter assays using HEK293T cells (EC50s = 0.94 and 1.5 μM, respectively) and is selective for these receptors over retinoic acid receptor α (RARα), retinoid X receptor α (RXRα), PPARα, PPARγ, and liver X receptor α (LXRα) at 10 μM.

Others

Others

2522515

C28H25Cl3N2O4

559.87

C(OC1=CC(Cl)=C(CNC2=CC=C(CC(O)=O)C=C2)C=C1)C=3C(=NOC3C(C)C)C4=C(Cl)C=CC=C4Cl

-20°C

Ice Packs

Small Compound