CB2R/5-HT1AR agonist 1 - CAS 2821085-76-9

Compound 2o, also known as CB2R/5-HT1AR agonist 1, serves as a partial orally active agonist for the CB2 receptor (EC50 = 479.6 nM) and a full agonist for the 5-HT1A receptor (EC50 = 2.7 μM) . This compound demonstrates both anti-anxiety and anti-depressive effects and has favorable pharmacokinetic properties [1].

Cannabinoid Receptor, 5-HT Receptor

Neuroscience, GPCR/G Protein

2821085-76-9

C24H33NO3

383.52

C(CCC)C1(CC1)C2=C(C(N)=O)C(O)=C(C(O)=C2)[C@H]3[C@H](C(C)=C)CCC(C)=C3

-20°C

Ice Packs

Small Compound