CB7993113 - CAS 819827-50-4

CB7993113 is a potent AHR antagonist with an IC50 of 0.33 μM, directly binding the AHR protein and blocking its nuclear translocation. It inhibits polycyclic aromatic hydrocarbon (PAH) - and TCDD-induced reporter activity by 75% and 90%, respectively [1].

Aryl Hydrocarbon Receptor

Immunology/Inflammation

819827-50-4

C15H10BrNO5

364.15

O(CC(N)=O)C1=C(OC=2C(C1=O)=CC=CC2)C=3OC(Br)=CC3

-20°C

Ice Packs

Small Compound