Molfinity

CCG-273220 - CAS 2750414-35-6

SKU:MF-0040397-01

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Product Details

Bioactivity
CCG-273220 is a covalent inhibitor of G protein-coupled receptor (GPCR) kinase 5 (GRK5) (IC50: 220 nM) .CCG-273220 covalently binds the GRK5 subfamily-specific residue Cys474 and is more selective for GRK5 than GRK2.
Target
Others, GRK
Related Pathways
GPCR/G Protein, Others
CAS Number
2750373
Molecular Formula
C26H24ClFN4O3
Molecular Weight
494.95
SMILES
C[C@@H](NC(=O)c1ccc2NC(=O)\C(=C/c3[nH]c(C)c(NC(=O)CCl)c3C)c2c1)c1ccc(F)cc1
Storage Temperature
-20°C
Shipping Conditions
Ice Packs
Category
Small Compound