CDK7/9-IN-1 - CAS 2747919-19-1

CDK7/9-IN-1 is a specific inhibitor of cyclin-dependent kinases 7/9 (CDK7/9), targeting CDK7 with IC50 values of 0.0656 μM without pre-incubation and 0.00574 μM after 3 hours pre-incubation, and displaying inhibitory activity against CDK9 with an IC50 of 2.14 μM after 3 hours pre-incubation, making it valuable for cancer research.

Others, CDK

Cell Cycle/Checkpoint, Others

2747899

C24H32F3N5O2

479.548

CC(C)c1cnc2c(NC3CCN(C[C@@H]4CN(CCO4)C(=O)C=C)CC3)cc(cn12)C(F)(F)F

-20°C

Ice Packs

Small Compound