Skip to product information
1 of 1

Molfinity

Cerlapirdine - CAS 925448-93-7

Cerlapirdine - CAS 925448-93-7

SKU:MF-0094674-01

Regular price $65.31 USD
Regular price Sale price $65.31 USD
Sale Sold out
Taxes included.
Size
Quantity
View full details
  • Bioactivity

    Cerlapirdine (PF-05212365) is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.

  • Target

    5-HT Receptor

  • Related Pathways

    GPCR/G Protein, Neuroscience

  • CAS Number

    925348

  • Purity

    0.9877

  • Molecular Formula

    C22H23N3O3S

  • Molecular Weight

    409.5

  • SMILES

    S(=O)(=O)(C=1C=2C(NN1)=CC=C(OCCCN(C)C)C2)C=3C4=C(C=CC3)C=CC=C4

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound