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CGP 57380 - CAS 522629-08-9
CGP 57380 - CAS 522629-08-9
SKU:MF-0006771-01
Regular price
$34.67 USD
Regular price
$21.45 USD
Sale price
$34.67 USD
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Product Details
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Bioactivity
CGP 57380 (MNK1 Inhibitor) is a potent MNK1 inhibitor with IC50 of 2.2 μM, exhibiting no inhibitory activity on p38, JNK1, ERK1 and -2, PKC, or c-Src-like kinases.
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Target
MNK, Apoptosis
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Related Pathways
Apoptosis, MAPK
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CAS Number
522629-08-9
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Purity
0.9989
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Molecular Formula
C11H9FN6
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Molecular Weight
244.23
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SMILES
Nc1ncnc2[nH]nc(Nc3ccc(F)cc3)c12
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Storage Temperature
-20°C
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Shipping Conditions
Ice Packs
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Category
Small Compound