CHF-6550 - CAS 3052116-62-5

CHF-6550 is an antagonist of the muscarinic M3 receptor (M3 receptor) and an agonist of the β2 adrenoceptor (β2 adrenoceptor), with pKi values of 9.3 and 10.6, respectively. It exhibits favorable hepatocyte clearance in rat models and demonstrates good pharmacokinetic properties in guinea pigs.

AChR, Adrenergic Receptor

GPCR/G Protein, Neuroscience

3052049

C42H46N4O8

734.84

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-20°C

Ice Packs

Small Compound