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CK2/ERK8-IN-1 - CAS 1085822-09-8

CK2/ERK8-IN-1 - CAS 1085822-09-8

MF-0021937-01

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Product Details

  • Bioactivity

    CK2/ERK8-IN-1 (TMCB) is a dual inhibitor of casein kinase 2 (CK2) (Ki: 0.25 μM) and ERK8 (IC50s: 0.50 μM) with pro-apoptotic efficacy. CK2/ERK8-IN-1 also binds to PIM1, DYRK1A, and HIPK2 (Kis: 8.65 μM, 11.9 μM, and 15.25 μM) .

  • Target

    DYRK, ERK, Pim, Apoptosis, Casein Kinase

  • Related Pathways

    Cell Cycle/Checkpoint, Tyrosine Kinase/Adaptors, Stem Cells, MAPK, JAK/STAT signaling, Apoptosis, Metabolism, Chromatin/Epigenetic

  • CAS Number

    1085822-09-8

  • Purity

    0.9882

  • Molecular Formula

    C11H9Br4N3O2

  • Molecular Weight

    534.82

  • SMILES

    CN(C)c1nc2c(Br)c(Br)c(Br)c(Br)c2n1CC(O)=O

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound