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CMPD101 - CAS 865608-11-3

CMPD101 - CAS 865608-11-3

MF-0019151-01

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Product Details

  • Bioactivity

    CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM) . Which can be used for the study of heart failure. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCα with IC50s of 3.1 μM , 2.3 μM, 1.4 μM and 8.1 μM, respectively.

  • Target

    PKC, GRK, ROCK

  • Related Pathways

    Cell Cycle/Checkpoint, Chromatin/Epigenetic, Stem Cells, GPCR/G Protein, Cytoskeletal Signaling

  • CAS Number

    865594

  • Purity

    0.9904

  • Molecular Formula

    C24H21F3N6O

  • Molecular Weight

    466.46

  • SMILES

    Cn1c(CNc2cccc(c2)C(=O)NCc2ccccc2C(F)(F)F)nnc1-c1ccncc1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound