CP-199331 - CAS 158102-93-3

CP-199331, a cysLT1 receptor antagonist, demonstrates equivalent potency to commercially available cysLT1 receptor antagonists zafirlukast and pranlukast. It shows favorable pharmacokinetic properties in both rats and monkeys, and unlike CP-85,958, no hepatotoxicity has been observed in monkeys.

158006

C26H21F5N2O6S2

616.58

O[C@H]1C=2C(OC[C@H]1CC3=C(OC)C=CC(NS(C(F)(F)F)(=O)=O)=C3)=CC=C(OCC4=NC=5C(S4)=CC(F)=C(F)C5)C2

-20°C

Ice Packs

Small Compound