CP94253 - CAS 131084-35-0

CP94253 is an orally active selective agonist of the serotonin receptor 1B (5-HT1B), exhibiting agonistic activity by competitively binding to 5-HT1 receptors with iodocyanopindolol (ICP) . It binds to the 5-HT1B, 5-HT1A, 5-HT1D, 5-HT1C, and 5-HT2 receptors with Ki values of 2, 89, 49, 860, and 1600 nM, respectively. In rat models, CP94253 induces satiety, anorexia, weight loss, and hyperactivity.

5-HT Receptor

Neuroscience, GPCR/G Protein

131084-35-0

C15H19N3O

257.33

N1=C(OCCC)C=CC=2NC=C(C12)C3=CCNCC3

-20°C

Ice Packs

Small Compound