CTAP - CAS 103429-32-9

Potent and selective μ opioid receptor antagonist (IC50 = 3.5 nM) . Displays > 1200-fold selectivity over δ opioid and somatostatin receptors. Brain penetrant and active in vivo.

Opioid Receptor

Endocrinology/Hormones, GPCR/G Protein, Neuroscience

103429-32-9

C51H69N13O11S2

1104.32

C[C@@H](O)[C@H](NC(=O)C1NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](CSSC1(C)C)NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(N)=O

-20°C

Ice Packs

Peptide