(D-Arg8) -Inotocin - CAS 745816-74-4

' (D-Arg8) -Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM. It demonstrates over 3000-fold selectivity for the human V1aR compared to the OTR, V1bR, and V2R subtypes [1].'

Vasopressin Receptor

GPCR/G Protein

745738

C39H68N14O11S2

973.17

C(=O)(N1[C@H](C(N[C@@H](C(NCC(N)=O)=O)CCCNC(=N)N)=O)CCC1)[C@H]2NC(=O)[C@H](CC(N)=O)NC(=O)[C@]([C@@H](C)O)(NC(=O)[C@]([C@H](CC)C)(NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)CSSC2)[H])[H]

-20°C

Ice Packs

Peptide