DCLK1-IN-2 - CAS 2978517-43-8

DCLK1-IN-2 (Compound I-5) is a potent inhibitor of DCLK1, exhibiting an IC50 of 171.3 nM, and demonstrates significant antiproliferative effects on SW1990 cell lines with an IC50 of 0.6 μM, as well as in vivo antitumor potency [1].

Others, Serine Protease

Others, Proteases/Proteasome

2978466

C26H32N8O3S

536.65

N(C1=C2C(=NC(NC3=C(OC)C=C(C=C3)N4CCN(C)CC4)=N1)N=CN2)C5=C(S(C(C)C)(=O)=O)C=CC=C5

-20°C

Ice Packs

Small Compound