Des-Gln14-Ghrelin - CAS 293735-04-3

An endogenous ligand for the ghrelin receptor (GHS-R1a), produced by alternative splicing of the rat ghrelin gene. Potently induces Ca2+ release in cells expressing ghrelin receptors (EC50 = 2.4 nM) and stimulates GH release in vivo.

GHSR

GPCR/G Protein

293735-04-3

C142H237N43O40

3186.7

C(=O)([C@H]1N(C([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CC2=CN=CN2)NC([C@@H](NC(=O)[C@H]3N(C([C@@H](NC([C@@H](NC([C@H](CC4=CC=CC=C4)NC([C@@H](NC([C@@H](NC(CN)=O)CO)=O)COC(CCCCCCC)=O)=O)=O)CC(C)C)=O)CO)=O)CCC3)CCC(O)=O)=O)=O)CCC(N)=O)=O)CCCCN)=O)C)=O)CCC(N)=O)=O)CCCNC(=N)N)=O)CCCCN)=O)CCC(O)=O)=O)CO)=O)CCCCN)=O)CCCCN)=O)CCC1)N5[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(=O)N6[C@H](C(N[C@@H](CCCNC(=N)N)C(O)=O)=O)CCC6)CCC(N)=O)=O)CC(C)C)=O)CCCCN)=O)C)=O)CCC5

-20°C

Ice Packs

Peptide