DHP-218 - CAS 102097-78-9

DHP-218 is a calcium channel antagonist. DHP-218 inhibits Calcium-induced contraction of the rat aorta in high K+ solution with the pA2 value of 9.11. The IC50 value for the inhibitory effects of DHP-218 in high K+-induced and phenylephrine-induced contraction are 6.3 nmol/l and 66 nmol/l respectively.

Others, Calcium Channel

Membrane transporter/Ion channel, Others, Metabolism

102010

C18H21N2O7P

408.34

C(OC)(=O)C=1C(C(=C(C)NC1C)P2(=O)OCCCO2)C3=C(N(=O)=O)C=CC=C3

-20°C

Ice Packs

Small Compound