Didesmethyl cariprazine - CAS 839712-25-3

Didesmethyl cariprazine, a metabolite of Cariprazine, is the major cyclic active part. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a potent D3 preference D3/D2 receptor partial agonist of dopamine for the treatment of schizophrenia, bipolar mania, and depression, with a high affinity for d3 and d2 receptors and a moderate affinity for 5-HT 1A receptors.

5-HT Receptor, Dopamine Receptor

Neuroscience, GPCR/G Protein

839684

0.997

C19H28Cl2N4O

399.36

NC(=O)N[C@H]1CC[C@H](CCN2CCN(CC2)c2cccc(Cl)c2Cl)CC1

-20°C

Ice Packs

Small Compound