DPP-4/GPR119 modulator 1 - CAS 2411099-68-6

DPP-4/GPR119 modulator 1 (Compound 22) is an orally active compound that acts as both a dipeptidyl peptidase IV (DPP-IV) inhibitor and GPR119 agonist, demonstrating a glucose-lowering effect in blood and moderate inhibition of the hERG channel with an IC50 value of 4.9 μM. This compound is applicable in diabetes research [1].

Potassium Channel, Proteasome, GPCR, Others

Others, Ubiquitination, GPCR/G Protein, Endocrinology/Hormones, Proteases/Proteasome, Membrane transporter/Ion channel

2411025

C30H39ClN10O3

623.15

Cl.CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nc(no3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1

-20°C

Ice Packs

Small Compound