EB1002 - CAS 2770688-48-5

EB1002 is a selective NK2R agonist that has demonstrated significant enhancements in the expression levels of genes associated with mitochondrial biogenesis (such as PGC-1α) in obese mice. This suggests that EB1002 promotes energy expenditure by enhancing mitochondrial activity. Additionally, EB1002 has improved insulin sensitivity and glucose-lipid metabolism in mice. Therefore, EB1002 holds potential for research into obesity and type 2 diabetes.

E3 Ligase Ligand-Linker Conjugate, Neurokinin receptor

Neuroscience, GPCR/G Protein, PROTAC

2770635

C73H124N12O23

1537.83

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-20°C

Ice Packs

Small Compound