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Echistatin - CAS 154303-05-6
Echistatin - CAS 154303-05-6
SKU:MF-0153293
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$1,436.45 USD
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$1,436.45 USD
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Product Details
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Bioactivity
Potent irreversible αVβ3 integrin antagonist (Ki = 0.27 nM) . Disrupts attachment of osteoclasts to bone and inhibits bone reabsorption (IC50 = 0.1 nM) . Prevents ADP-induced platelet aggregation via inhibition of glycoprotein IIb/IIIa (GpIIb/IIIa, αIIbβ3) receptors (IC50 = 30 nM) in vitro.
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Target
Integrin
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Related Pathways
Cytoskeletal Signaling
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CAS Number
154303-05-6
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Molecular Formula
C217H341N71O74S9
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Molecular Weight
5417.1
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Storage Temperature
-20°C
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Shipping Conditions
Ice Packs
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Category
Peptide