ELA-11 (human) - CAS 1784687-32-6

High affinity apelin receptor agonist (Ki = 14 nM) . Bioactive fragment of ELA-32. Inhibits forskolin-induced cAMP production and stimulates β-arrestin recruitment in vitro.

Apelin receptor, Arrestin

GPCR/G Protein

1784649

C58H90N16O13S2

1283.57

C(N[C@H](C(=O)N1[C@H](C(O)=O)CCC1)CC2=CC=CC=C2)(=O)[C@H]3N(C([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CC4=CN=CN4)NC([C@@H](NC(=O)[C@H]5N(C([C@@H](NC([C@H](CS)N)=O)CCSC)=O)CCC5)CC(C)C)=O)=O)CO)=O)CCCNC(=N)N)=O)[C@@H](C)C)=O)CCC3

-20°C

Ice Packs

Peptide