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EP4 receptor antagonist 1 - CAS 2287259-07-6

EP4 receptor antagonist 1 - CAS 2287259-07-6

MF-0022239-01

$111.94 USD
$111.94 USD
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Product Details

  • Bioactivity

    EP4 Receptor Antagonist 1 is a highly potent and selective competitive prostanoid EP4 receptor antagonist, effective for cancer immunotherapy. It inhibits both human and mouse EP4 receptors with IC50 values of 6.1 nM and 16.2 nM, respectively, while displaying minimal activity (IC50s >10 μM) against human EP1, EP2, and EP3 receptors.

  • Target

    Prostaglandin Receptor

  • Related Pathways

    Immunology/Inflammation, GPCR/G Protein

  • CAS Number

    2287259-07-6

  • Purity

    0.9953

  • Molecular Formula

    C23H21F3N4O3

  • Molecular Weight

    458.43

  • SMILES

    C\C=C\c1nnn(Cc2ccc(cc2)C(F)(F)F)c1C(=O)N[C@@H](C)c1ccc(cc1)C(O)=O

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound