EPI-7170 - CAS 2139288-26-7

EPI-7170 is a ralaniten analogue and a potent antagonist of the androgen receptor N-terminal structural domain, blocking the transcriptional activity of the full-length AR (FL-AR) and AR splice variants (AR-Vs) . EPI-7170 exhibits antitumor activity against enzalutamide resistant debulking resistant prostate cancer (CRPC) .

Others, Androgen Receptor

Others, Endocrinology/Hormones

2139255

C22H28Cl3NO6S

540.88

C(C)(C)(C1=CC(Cl)=C(OC[C@@H](CCl)O)C(Cl)=C1)C2=CC=C(OC[C@@H](CNS(C)(=O)=O)O)C=C2

-20°C

Ice Packs

Small Compound