EPZ-719 - CAS 2697176-16-0

EPZ-719 is a highly selective and potent inhibitor of SETD2, a novel compound known for its ability to inhibit the enzymatic activity of SETD2 (IC50 = 0.005 μM) . This compound displays a remarkable selectivity over other histone methyltransferases, making it a promising candidate for targeted therapeutic applications in the field of epigenetic research.

Histone Methyltransferase, Others

Chromatin/Epigenetic, Others

2697160

C22H31FN4O3S

450.57

CN([C@H]1CCN(C1)[C@H]1CCC[C@H](C1)NC(=O)c1cc2c(F)ccc(C)c2[nH]1)S(C)(=O)=O

-20°C

Ice Packs

Small Compound