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Molfinity

EZH2-IN-14 - CAS 1979157-17-9

EZH2-IN-14 - CAS 1979157-17-9

MF-0146549-01

$1,778.67 USD
$1,778.67 USD
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Product Details

  • Bioactivity

    EZH2-IN-14 is a selective inhibitor of EZH2 (Histone Methyltransferase) with an IC50 value of 12 nM, targeting the methyltransferase activity of EZH2/PRC2 and reducing H3K27me3 levels. It exhibits more than 200-fold selectivity for EZH2 over the closely related H3K27 methyltransferase, EZH1.

  • Target

    Histone Methyltransferase, Others

  • Related Pathways

    Chromatin/Epigenetic, Others

  • CAS Number

    1979131

  • Molecular Formula

    C31H39N7O2

  • Molecular Weight

    541.69

  • SMILES

    C(C)(C)N1C=2C(=C(C(NCC3=C(C)C=C(C)NC3=O)=O)C=C(C2)C=4C=CC(=NC4)N5CCN(C(C)C)CC5)C=N1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound