Fiduxosin - CAS 208993-54-8

Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with Ki values of 0.160 nM, 24.9 nM and 0.920 nM, respectively. Fiduxosin can be used for the treatment of benign prostatic hyperplasia.

Adrenergic Receptor

GPCR/G Protein, Neuroscience

208931

0.9973

C30H29N5O4S

555.65

O=C1C2=C(C=3C(S2)=NC=C(N3)C4=CC=CC=C4)NC(=O)N1CCCCN5C[C@@]6([C@](C5)(COC=7C6=C(OC)C=CC7)[H])[H]

-20°C

Ice Packs

Small Compound