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Molfinity

Firibastat - CAS 648927-86-0

Firibastat - CAS 648927-86-0

MF-0039259-01

$40.65 USD
$40.65 USD
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Product Details

  • Bioactivity

    Firibastat (RB150) is a glutamyl aminopeptidase antagonist and an orally active brain penetrating prodrug of EC33. It is a first-in-class brain aminopeptidase A (APA) inhibitor with a Ki of 200 nM. Firibastat selectively and specifically inhibits conversion of brain angiotensin-II into angiotensin-III and decreases blood pressure in hypertensive rats[1][2].

  • Target

    Aminopeptidase

  • Related Pathways

    Metabolism

  • CAS Number

    648841

  • Purity

    0.9988

  • Molecular Formula

    C8H20N2O6S4

  • Molecular Weight

    368.51

  • SMILES

    N[C@@H](CCS(O)(=O)=O)CSSC[C@@H](N)CCS(O)(=O)=O

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound