FLTX1 - CAS 1481401-71-1

FLTX1 is a fluorescent derivative of Tamoxifen, designed to efficiently target and label intracellular Tamoxifen-binding sites (estrogen receptors) both under permeabilized and non-permeabilized conditions. Additionally, FLTX1 demonstrates strong antiestrogenic activity in breast cancer cells, resembling the potent antiestrogenic properties of Tamoxifen. Notably, FLTX1 does not exhibit any estrogenic agonistic effect on the uterus.

Estrogen/progestogen Receptor, Estrogen Receptor/ERR

Endocrinology/Hormones

1481401-71-1

0.9846

C31H28N4O4

520.58

C(=C(/CC)\C1=CC=CC=C1)(\C2=CC=C(OCCN(C)C=3C=4C(C(N(=O)=O)=CC3)=NON4)C=C2)/C5=CC=CC=C5

-20°C

Ice Packs

Small Compound