FT001 - CAS 1778655-51-8

FT001 is a potent, selective and orally available inhibitor of BET Bromodomain with antitumor activity. FT001 inhibited the expression of MYC with the IC50 value of 0.46 μM) . FT001 has potent antiproliferative effects against MV-4-11 and demonstrates significant MYC mRNA suppression both in vitro and in vivo.

Epigenetic Reader Domain

Chromatin/Epigenetic

1778596

>99.99%

C25H29N3O4S

467.58

C(=O)(N1C=2C(N(C(C)=O)[C@@H](C)C1)=CC=C(C2)C3=CC=C(C=C3)N4CCS(=O)(=O)CC4)C5CC5

-20°C

Ice Packs

Small Compound