Gemigliptin tartrate hydrate - CAS 1375415-82-9

Gemigliptin (LC15-0444) tartrate hydrate is a selective, reversible, and competitive inhibitor of dipeptidyl peptidase 4 (DPP-4), with an IC50 value of 10.3 nM for human recombinant DPP-4. It exhibits strong anti-glycation properties and is used in research on advanced glycation end product-related diabetic complications.

Proteasome

Proteases/Proteasome, Ubiquitination

1375324

C22H27F8N5O9

657.47

[C@@H]([C@H](C(O)=O)O)(C(O)=O)O.C(F)(F)(F)C1=C2C(CN(C(C[C@@H](CN3CC(F)(F)CCC3=O)N)=O)CC2)=NC(C(F)(F)F)=N1.O

-20°C

Ice Packs

Small Compound