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Molfinity

GI-530159 - CAS 69563-88-8

GI-530159 - CAS 69563-88-8

MF-0040154-01

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Product Details

  • Bioactivity

    TREK1 and TREK2 channel activator (EC50 = 0.76 μM in Rb efflux assay in TREK1-expressing CHO cells) . Exhibits selectivity for TREK1/2 over TRAAK, TASK3 and a range of other potassium channels. Hyperpolarizes membrane potential of dorsal root ganglion neurons and depresses neuronal activity in vitro.

  • Target

    Others, Potassium Channel

  • Related Pathways

    Membrane transporter/Ion channel, Others

  • CAS Number

    69467

  • Molecular Formula

    C27H20F6N2O2

  • Molecular Weight

    518.45

  • SMILES

    Nc1ccc(Oc2ccc(cc2)C(c2ccc(Oc3ccc(N)cc3)cc2)(C(F)(F)F)C(F)(F)F)cc1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound